Ibodutant;化合物 T16039MEN 15596;MEN 15596 (2024/9/1)
简介:ibodutant is an effective and selective tachykinin nk2 receptor antagonist (pki: 10.1).
Men 10376;化合物 T16038Neurokinin-2 receptor antagonist;Neurokinin-2 receptor antagonist (2024/9/1)
简介:men 10376 is a selective antagonist of tachykinin nk-2 receptor. it has a ki of 4.4 μm for rat small intestine nk-2 receptor.
GLN-1062;化合物GLN-1062GLN-1062 (2024/9/1)
简介:gln-1062 is a pro-drug of galantamine and liberates galantamine on cleavage by a carboxyesterase in the brain.
Melinamide;甲亚油酰胺AC 223|||DL-N-(α-Methylbenzyl)linoleamide;甲亚油酰胺|||AC 223|||DL-N-(α-Methylbenzyl)lino (2024/9/1)
简介:melinamide is an amide derivative of an unsaturated long-chain fatty acid and also is an inhibitor of cholesterol absorption (ic50: 20.9 μm).
Meleagrin;化合物 T16035Meleagrin (2024/9/1)
简介:meleagrin, a roquefortine c-derived alkaloid produced by penicillium fungi, serves as both a class of fabi inhibitors and a lead c-met inhibitory entity for controlling c-met-dependent metastatic and invasive breast malignancies. it exhibits antimicrobial and anti-proliferative activities.
血站恒温振荡保存设备 (2024/9/1)
简介:血站恒温振荡保存设备高效保温:采用先进的保温技术,能够有效保持血小板的温度稳定,确保在长时间内维持血小板的适宜温度,保障其质量和活性。精确控温:配备精确的温度控制系统,用户可以根据需要精确调节保存温度,以满足不同血小板的保存要求。控温范围通常为22.0℃±2.0℃,确保血小板在佳保存温度范围内。
Meclinertant;化合物 T16034SR 48692;SR 48692 (2024/9/1)
简介:meclinertant is an effective, selective, nonpeptide, and orally active neurotensin receptor 1 (nts1) antagonist. meclinertant competitively antagonizes neurotensin-induced intracellular ca2+ mobilization (pa2 : 8.13), in human colon carcinoma (ht-29) cells. meclinertant has anxiolytic, anti-addictive, and memory-impairing effects.
ME1111;化合物ME1111ME1111 (2024/9/1)
简介:me1111, a succinate dehydrogenase inhibitor of trichophyton species, serves as an antifungal agent effective against dermatophytes. notably proficient in penetrating human nails, it is utilized in onychomycosis research.
中心血站恒温振荡保存箱 (2024/9/1)
简介:中心血站恒温振荡保存箱高效保温:采用先进的保温技术,能够有效保持血小板的温度稳定,确保在长时间内维持血小板的适宜温度,保障其质量和活性。精确控温:配备精确的温度控制系统,用户可以根据需要精确调节保存温度,以满足不同血小板的保存要求。控温范围通常为22.0℃±2.0℃,确保血小板在佳保存温度范围内。
(Z)-MDL 105519;异构体MDL 105519(Z)-MDL 105519 (2024/9/1)
简介:(z)-mdl 105519 is an inactive isomer of mdl105519.
MDL 105519;化合物 T16032MDL 105519 (2024/9/1)
简介:mdl 105519 is an effective antagonist of glycine binding to the nmda receptor.
McMMAF;化合物McMMAFMaleimidocaproyl monomethylauristatin F;Maleimidocaproyl monomethylauristatin F (2024/9/1)
简介:mcmmaf is a protective group-conjugated mmaf. mmaf is a potent tubulin polymerization inhibitor.it is a mmaf derivative having a maleimidocaproyl linker (mc linker), which is ready to conjugate to antibody or other proteins or biopolymers. mafodotin is a useful agent for make antibody drug conjugate (adc) for targeted drug delivery.
Mcl1-IN-8;化合物 T16030Mcl1-IN-8 (2024/9/1)
简介:mcl1-in-8 is an mcl-1-puma interface inhibitor (ki: 0.3 μm). in cancer cells, mcl1-in-8 shows dual activity on reducing puma-dependent apoptosis while deactivating mcl-1-mediated anti-apoptosis.
Glipizide格列吡嗪CP 28720|||K 4024|||格列吡嗪 (2024/9/1)
简介:glipizide (cp 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.
Mcl1-IN-3;化合物 T16029Mcl1-IN-3 (2024/9/1)
简介:mcl1-in-3 is an mcl1 inhibitor. it has an ic50 and ki of 0.67 and 0.13 μm, respectively.
IMB-XH1;7-[(2-吡啶基氨基)-2-噻吩基甲基]-8-喹啉醇Mcl1-IN-2;Mcl1-IN-2|||7-[(2-吡啶基氨基)-2-噻吩基甲基]-8-喹啉醇 (2024/9/1)
简介:imb-xh1 (mcl1-in-2) is a myeloid cell factor 1 (mcl-1) inhibitor.
Mcl1-IN-1;化合物 T16027Mcl1-IN-1 (2024/9/1)
简介:mcl1-in-1 is a myeloid cell factor 1 inhibitor (ic50=2.4 μm).
MCI826;化合物MCI826MCI826 (2024/9/1)
简介:mci826 is a potent and selective antagonist of p-glycoprotein (p-gp) and peptide leukotrienes (p-lts), showing anti-asthmatic activity in a guinea pig model of advanced asthma.
SGD-1910;化合物 T16025MC-Val-Ala-PBD;MC-Val-Ala-PBD (2024/9/1)
简介:mc-val-ala-pbd is a drug-linker conjugate for adc by using the antitumor antibiotic, pyrrolobenzodiazepine (pbd, a cytotoxic dna crosslinking), linked via the cleavable linker mc-val-ala[1].
血液中心振荡保存箱 (2024/9/1)
简介:血液中心振荡保存箱高效保温:采用先进的保温技术,能够有效保持血小板的温度稳定,确保在长时间内维持血小板的适宜温度,保障其质量和活性。精确控温:配备精确的温度控制系统,用户可以根据需要精确调节保存温度,以满足不同血小板的保存要求。控温范围通常为22.0℃±2.0℃,确保血小板在佳保存温度范围内。
MC-GGFG-DX8951;化合物 T16024MC-GGFG-DX8951 (2024/9/1)
简介:mc-ggfg-dx8951 is a drug-linker conjugate designed for antibody-drug conjugation (adc) that demonstrates antitumor activity through the deployment of dx8951, a dna topoisomerase i inhibitor, connected using the protease-cleavable mc-ggfg linker[1].
(24S)-MC 976;化合物 T16023L2(24S)-MC 976 (2024/9/1)
简介:(24s)-mc 976 is a derivative of vitamin d3.
(24R)-MC 976;化合物 T16023L(24R)-MC 976 (2024/9/1)
简介:(24r)-mc 976 is a derivative of vitamin d3.
MC 976;化合物 T16023MC 976 (2024/9/1)
简介:mc 976 is a derivative of vitamin d3.
MBQ-167;化合物MBQ-167MBQ-167 (2024/9/1)
简介:mbq-167 is a dual inhibitor of rac/cdc42 (ic50s: 103 nm for rac 1/2/3 and 78 nm for cdc42 in mda-mb-231 cells, respectively).
Valproic acid sodium salt;丙戊酸钠Sodium Valproate;丙戊酸钠|||Sodium Valproate (2024/9/1)
简介:valproic acid sodium salt (sodium valproate) is the sodium salt form of valproic acid with anti-epileptic activity. valproic acid sodium salt is converted into its active form, valproate ion, in blood. although the mechanism of action remains to be elucidated, valproic acid sodium salt increases concentrations of gamma-aminobutyric acid (gaba) in the brain, probably due to inhibition of the enzymes responsible for the catabolism of gaba. this potentiates the synaptic actions of gaba. valproic ac
MB-7133;化合物 T16019MB-7133 (2024/9/1)
简介:mb-7133 is an inhibitor of dna synthesis.
MB-07811;化合物MB-07811VK-2809;VK-2809 (2024/9/1)
简介:mb-07811 (vk-2809) is an orally active hepdirect prodrug of mb07344 with cholesterol and triglycerides lowering activity. mb-07811 is an agonist of liver-targeted thr-β.
Maytansinol;美登醇Ansamitocin P-0;美登醇|||Ansamitocin P-0 (2024/9/1)
简介:maytansinol (ansamitocin p-0) inhibits microtubule assembly and causes microtubule disassembly in vitro.
Maxacalcitol;马沙骨化醇22-Oxacalcitriol;马沙骨化醇|||22-Oxacalcitriol (2024/9/1)
简介:maxacalcitol (22-oxacalcitriol) is a ligand of vdr-like receptors and a non-serum calcium vitamin d3 analogue. maxacalcitol inhibits parathyroid hormone (pth) mrna expression in vitro and in vivo.