9月
保存血小板的恒温振荡设备 (2024/9/1)
简介：保存血小板的恒温振荡设备高效保温：采用先进的保温技术，能够有效保持血小板的温度稳定，确保在长时间内维持血小板的适宜温度，保障其质量和活性。精确控温：配备精确的温度控制系统，用户可以根据需要精确调节保存温度，以满足不同血小板的保存要求。控温范围通常为22.0℃±2.0℃，确保血小板在佳保存温度范围内。
MAT2A inhibitor 1；化合物 T16013MAT2A inhibitor 1 (2024/9/1)
简介：mat2a inhibitor 1 is an inhibitor of methionine adenosyltransferase 2a (mata2) (ic50 < l00 nm).
Marizomib；马里佐米NPI-0052|||Salinosporamide A|||ML858；NPI-0052|||Salinosporamide A|||ML858 (2024/9/1)
简介：marizomib (ml858) is a novel irreversible brain-permeable proteasome inhibitor that inhibits ct-l (β5), ct-t-laspase-like (c-l, β1), and trypsin-like (t-l, β2) 20s proteasomes with ic50s of 3.5, 28, and 430 nm, respectively.
Manumycin A；手霉素AManumycin A (2024/9/1)
简介：manumycin a is an antibiotic. manumycin a induces apoptosis and exerts antitumor activity. manumycin a inhibits exosome biogenesis and secretion via targeted inhibition of ras/raf/erk1/2 signaling. manumycin a acts as a selective, competitive inhibitor of protein farnesyltransferase (ftase) with respect to farnesylpyrophosphate (ki =1.2 μm), and as a noncompetitive inhibitor with respect to the ras protein.
Mancozeb；代森锰锌Mancozeb (2024/9/1)
简介：mancozeb is a fungicide of ethylene-bis-dithiocarbamate.
Lomustine；洛莫司汀CCNU|||NSC 79037；CCNU|||NSC 79037|||洛莫司汀 (2024/9/1)
简介：lomustine (nsc-79037) is an alkylating agent of value against both hematologic malignancies and solid tumors.
医用恒温振荡保存箱 (2024/9/1)
简介：医用恒温振荡保存箱高效保温：采用先进的保温技术，能够有效保持血小板的温度稳定，确保在长时间内维持血小板的适宜温度，保障其质量和活性。精确控温：配备精确的温度控制系统，用户可以根据需要精确调节保存温度，以满足不同血小板的保存要求。控温范围通常为22.0℃±2.0℃，确保血小板在佳保存温度范围内。
Managlinat dialanetil；地马格列MB06322|||MB 6322|||CS-917；MB06322|||MB 6322|||CS-917 (2024/9/1)
简介：managlinat dialanetil (mb06322) is an orally available and potent fructose 1,6-bisphosphatase (fbpase) inhibitor with hypoglycaemic activity for the study of type 2 diabetes.
输血科恒温振荡保存箱 (2024/9/1)
简介：输血科恒温振荡保存箱高效保温：采用先进的保温技术，能够有效保持血小板的温度稳定，确保在长时间内维持血小板的适宜温度，保障其质量和活性。精确控温：配备精确的温度控制系统，用户可以根据需要精确调节保存温度，以满足不同血小板的保存要求。控温范围通常为22.0℃±2.0℃，确保血小板在佳保存温度范围内。
Maleimido-tri(ethylene glycol)-propionic acid；化合物 T16008Mal-PEG3-acid；Mal-PEG3-acid (2024/9/1)
简介：maleimido-tri(ethylene glycol)-propionic acid is a cleavable adc linker used in the synthesis of antibody-drug conjugates (adcs). maleimido-tri(ethylene glycol)-propionic acid is used for the preparation of neolymphostin-based adc precursors for site-specific cysteine mutant trastuzumab-a114c conjugation[1].
MALAT1-IN-1；化合物MALAT1-IN-1MALAT1-IN-1 (2024/9/1)
简介：malat1-in-1 modulated malat1 downstream genes in a dose-dependent manner without affecting the expression of nuclear enriched abundant transcript 1 (neat1). malat1-in-1 is an effective and specific malat1 inhibitor.
Mal-Sulfo-DBCO；化合物 T16006Mal-Sulfo-DBCO (2024/9/1)
简介：mal-sulfo-dbco serves as a cleavable linker for the synthesis of antibody-drug conjugates (adcs)[1].
CDK2-IN-4；化合物CDK2-IN-4CDK2-IN-4 (2024/9/1)
简介：cdk2-in-4 is a potent and selective inhibitor of cdk2 with an ic50 of 44 nm for cdk2/cyclin a. it shows 2,000-fold selectivity over cdk1/cyclin b with ic50 of 86 um.
CDK12-IN-E9；化合物 T14915CDK12-IN-E9 (2024/9/1)
简介：cdk12-in-e9 is a potent and selective covalent cdk12 inhibitor and non-covalent cdk9 inhibitor while avoiding abc transporter-mediated efflux. it has a weak binding ability to cdk7/cyclinh complex (ic50> 1 μm).
Cdk1/2 Inhibitor III；Cdk1/2 抑制剂IIICdk1/2 Inhibitor III (2024/9/1)
简介：cdk1/2 inhibitor iii is a selective cdk1/2 inhibitor with an ic50 value of 2.1 μm against cdk1/cyclin b.
CD38 inhibitor 1；化合物CD38 inhibitor 1CD38 inhibitor 1 (2024/9/1)
简介：cd38 inhibitor 1 is an inhibitor of cd38. for hcd38 and mouse cd38, the ic50s are 7.3 nm and 1.9 nm.
CD3254；化合物CD3254CD3254 (2024/9/1)
简介：cd3254 is a selective and potent retinoid x receptor-like (rxr) agonist that inhibits neuronal cell death with ogd/reoxygenation.
CD2665；化合物CD2665CD2665 (2024/9/1)
简介：cd2665 is an orally active antagonist of retinoic acid receptor (rar). for rarγ and rarβ, the kis are 110 nm and 306 nm.
CD161；化合物 T14910NKR-P1A；NKR-P1A (2024/9/1)
简介：cd161 is a potent, selective, and orally bioavailable bet bromodomain inhibitor (ic50s: 28.2 nm and 7.2 nm for brd4 bd1 and brd4 bd2) with good anticancer activity.
Atovaquone；阿托伐醌Atavaquone；Atavaquone|||阿托伐醌 (2024/9/1)
简介：atovaquone (atavaquone) is a hydroxynaphthoquinone that has antimicrobial activity and is being used in antimalarial protocols.
CCX140；化合物CCX140CCX140-B；3-三氟甲基-4-氯-N-[2-[7H-吡咯并[2,3-D]嘧啶-4-羰基]-5-甲基-3-吡啶基]苯磺酰胺|||CCX140-B (2024/9/1)
简介：ccx140 (ccx140-b) (ccx140-b) is an antagonist of ccr2.
CCT367766；化合物CCT367766CCT367766 (2024/9/1)
简介：cct367766 is a potent, protac-based, third-generation, iso-functional pirin-targeted protein degradation probe (pdp) that depletes pirin expression at low concentrations.cct367766 has an ic50 value of 490 nm for the crbn-ddb1 complex.cct367766 has a good affinity for recombinant pirin and crbn. cct367766 has a good affinity for recombinant pirin and crbn, with kd values of 55 nm and 120 nm, respectively. cct367766 is a potent orally active protein that reduces the expression of pirin at low conc
CCT251545；化合物CCT251545CCT251545 (2024/9/1)
简介：cct251545 is an potent and oral-bioavailable wnt signaling inhibitor(ic50 of 5 nm in 7df3 cells).
CCT251455；化合物 T14906CCT251455 (2024/9/1)
简介：cct251455 is an inhibitor of mitotic kinase monopolar spindle 1 (mps1; ic50: 3 nm).
CCT251236；化合物 CCT251236CCT251236 (2024/9/1)
简介：cct251236 is a cell-based phenotypic high-throughput screening (hts) chemical probe developed to screen for inhibitors of the hsf1 stress pathway.cct251236 exhibits antimyeloma activity and inhibits hsf1.
CCT244747；化合物 T14904CCT244747 (2024/9/1)
简介：cct244747 is a chk1 inhibitor (ic50: 7.7 nm) and also abrogates g2 checkpoint (ic50: 29 nm).
CCT129957；化合物CCT129957CCT129957 (2024/9/1)
简介：cct129957 is a novel and potent phospholipase c-γ (plc-γ) inhibitor with an ic50 of about 3 μm and a gc50 of 15 μm.cct129957 exhibits anticancer activity and inhibits ca2+ release in squamous cells.
CCT020312；化合物CCT020312CCT020312 (2024/9/1)
简介：cct020312 is a selective activator of eif2ak3 and perk. cct020312 durably inhibits cell proliferation and elicits the phosphorylation of eif2a.
CCT-251921；化合物CCT-251921CCT-251921 (2024/9/1)
简介：cct-251921 is a potent, selective, and orally bioavailable cdk8 inhibitor (ic50: 2.3 nm).
CCR2-RA-[R]化合物CCR2-RA-[R](5R)-4-乙酰基-1-(4-氯-2-氟苯基)-5-环己基-1,5-二氢-3-羟基-2H-吡咯-2-酮 (2024/9/1)
简介：ccr2-ra-[r] is a c-c chemokine receptor type 2 (ccr2) allosteric antagonist (ic50: 103 nm).
MSN交谈
