9月
Risdiplam；化合物RisdiplamRO7034067|||RG7916；RO7034067|||RG7916 (2024/9/1)
简介：risdiplam (ro7034067) (rg7916) is orally administered. risdiplam is a centrally and peripherally distributed smn2 pre-mrna splicing modifier which increases survival motor neuron (smn) protein levels[1].
Risarestat；利沙司他CT 112；CT 112 (2024/9/1)
简介：risarestat (ct-112) is a potent aldose reductase inhibitor and thyroid hormone receptor (tr) antagonist for the treatment of hypoglycemia.
RIPK-IN-4；化合物 T16755RIPK-IN-4 (2024/9/1)
简介：ripk-in-4 is an effective and selective inhibitor of ripk2. it also has excellent oral bioavailability (ic50: 3 nm).
RIPGBM；化合物RIPGBMRIPGBM (2024/9/1)
简介：ripgbm is a selective inducer of apoptosis in glioblastoma multiforme cancer stem cells (ec50: ≤500 nm).
RIP2 kinase inhibitor 2；化合物 T16753RIP2 kinase inhibitor 2 (2024/9/1)
简介：rip2 kinase inhibitor 2 is a receptor-interacting protein-2 kinase inhibitor.
Rimacalib化合物 T16752SMP 114 (2024/9/1)
简介：rimacalib is an inhibitor of ca2+/calmodulin-dependent protein kinase ii (ic50s: ~1 μm for camkiiα and ~30 μm for camkiiγ).
Rilapladib；瑞拉帕地SB 659032；SB 659032 (2024/9/1)
简介：rilapladib (sb 659032) is a selective inhibitor of lipoprotein-associated phospholipase a2(lp-pla2, ic50 = 230 pm) and an antagonist of the platelet activating factor receptor.
Rigosertib；瑞格色替ON-01910；ON-01910|||瑞格色替 (2024/9/1)
简介：rigosertib (on-01910) is a selective and non-atp-competitive inhibitor of plk1 (ic50: 9 nm). rigosertib is a multi-kinase inhibitor and a selective anti-cancer agent, which induces apoptosis by inhibition of the pi3 kinase/akt pathway, promotes the phosphorylation of histone h2ax and induces g2/m arrest in the cell cycle.
Adefovir dipivoxil；阿德福韦酯Hepsera|||GS 0840|||Preveon；Hepsera|||GS 0840|||阿德福韦酯|||Preveon (2024/9/1)
简介：adefovir dipivoxil (gs 0840) is a dipivoxil formulation of adefovir, a nucleoside reverse transcriptase inhibitor analog of adenosine with activity against hepatitis b virus (hbv), herpes virus, and human immunodeficiency virus (hiv).
Rifalazil；利福拉齐KRM-1648|||ABI-1648；利福拉齐|||KRM-1648|||ABI-1648 (2024/9/1)
简介：rifalazil is a rifamycin derivative, inhibits the bacterial dna-dependent rna polymerase and kills bacterial cells by blocking off the β-subunit in rna polymerase. rifalazil is an antibiotic, exhibits high potency against mycobacteria, gram-positive bacteria, helicobacter pylori, c. pneumoniae and c. trachomatis (mic: 0.00025 to 0.0025 μg/ml).
Ridinilazole；化合物RidinilazoleSMT19969；SMT19969 (2024/9/1)
简介：ridinilazole (smt19969) is a novel narrow-spectrum nonabsorbable antibiotic. ridinilazole showed potent inhibition of c. difficile (mic90=0.125 mg/l) and was markedly more active than either metronidazole (mic90 = 8 mg/l) or vancomycin (mic90 = 2 mg/l).
Riboflavin Tetrabutyrate；四丁酸核糖黄素酯Riboflavin Tetrabutyrate (2024/9/1)
简介：riboflavin tetrabutyrate is a lipophilic flavin derivative. riboflavin tetrabutyrate has antioxidative and lipid peroxide-removing activity.
Rhosin；化合物 T16746Rhosin (2024/9/1)
简介：rhosin is an effective and specific rhoa subfamily rho gtpases inhibitor, which specifically binds to rhoa to inhibit rhoa-gef interaction (kd: ~ 0.4 um). rhosin does not interact with cdc42 or rac1, nor the gef, larg. rhosin causes cell apoptosis.
Rhosin hydrochloride；化合物Rhosin hydrochlorideRhosin hydrochloride (2024/9/1)
简介：rhosin hydrochloride is an effective and specific rhoa subfamily rho gtpases inhibitor, which specifically binds to rhoa to inhibit rhoa-gef interaction (kd: ~ 0.4 um). rhosin hydrochloride does not interact with cdc42 or rac1, nor the gef, larg. rhosin hydrochloride causes cell apoptosis.
Rhodamine 6G罗丹明6GBasic Red 1|||罗丹明6G|||罗丹明 6G (2024/9/1)
简介：rhodamine 6g (basic red 1) is a rhodamine analog useful in pgp efflux assays. it can be widely used in characterizing the kinetics of mrp1- mediated efflux as a laser dye and potential mitochondrial probe.
Rhodamine 123 free base；化合物 T16743LRhodamine 123 free base (2024/9/1)
简介：the laser dye rhodamine 123 inhibit mitochondrion function.
Rhodamine 123；罗丹明123R-22420|||RH-123；R-22420|||罗丹明 123|||RH-123|||罗丹明123 (2024/9/1)
简介：rhodamine 123 is a fluorescent dye (λex=503 nm, λem=527 nm).
Rhodamine 110；罗丹明110Rhodamine 110 chloride|||RH110；Rhodamine 110 chloride|||RH110|||罗丹明110 (2024/9/1)
简介：rhodamine 110 (rh110) is a xanthene dye similar to fluorescein and eosin.
Rheb inhibitor NR1Rheb 抑制剂 NR1Rheb inhibitor NR1|||Rheb inhibitor NR-1 (2024/9/1)
简介：rheb inhibitor nr1 is a rheb inhibitor and selective mtorc1 inhibitor.rheb inhibitor nr1 inhibits the phosphorylation of t389ps6k1 and promotes the phosphorylation of s473pakt.
RH1；化合物 RH1NSC 697726；NSC 697726 (2024/9/1)
简介：rh1 (nsc 697726) is a bioreductive anticancer compound that exhibits dose-dependent biphasic effects in vitro, inducing apoptosis at higher doses and senescence at lower doses.
Nateglinide；那格列奈A4166|||Senaglinide；那格列奈|||A4166|||Senaglinide (2024/9/1)
简介：nateglinide (senaglinide) is an oral hypoglycemic agent and amino acid derivative that stimulates insulin secretion from the pancreas and is used in the therapy of type 2 diabetes. nateglinide has been linked to rare instances of clinically apparent acute liver injury.
RG-12525；化合物RG-12525NID 525；NID 525 (2024/9/1)
简介：rg-12525（nid 525） is an orally available, selective and competitive leukotriene d (ltd) antagonist that inhibits ltc4, ltd4 and lte4-induced contraction of guinea pig thin-walled bands, with ic50 values of 2.6 nm, 2.5 nm, and 7 nm, respectively.rg-12525 inhibits cyp3a4, with a ki value of 0.5 µm. rg-12525 is a novel and potent ppar-γ agonist (ic50 value of about 60 nm) with species specificity for the study of asthma.
RF9 acetate；化合物RF9 acetateRF9 acetate (2024/9/1)
简介：rf9 acetate is an effective and selective antagonist of neuropeptide ff receptor with ki values of 58 and 75 nm for hnpff1r and hnpff2r, respectively.
RF9化合物 T16738RF9|||RF-9 (2024/9/1)
简介：rf9 is an effective and selective antagonist of the neuropeptide ff receptor (kis: 58±5 and 75±9 nm for hnpff1r and hnpff2r, respectively).
Revexepride；化合物 T16737Revexepride (2024/9/1)
简介：revexepride is a highly selective agonist of the 5-ht4 receptor and a potential inducer of cyp3a4 enzyme. revexepride is used for the treatment of gastroesophageal reflux disease.
Retosiban；化合物 T16736GSK 221149|||GSK 221149A；GSK 221149|||GSK 221149A (2024/9/1)
简介：retosiban is an effective and selective oxytocin antagonist (ki: 0.65 nm).
RET-IN-1；化合物 T16735RET-IN-1 (2024/9/1)
简介：ret-in-1 is a ret kinase inhibitor (ic50s: 1 nm, 7 nm, and 101 nm for ret (wt), ret (v804m) , and ret (g810r), respectively).
Resorufin sodium salt；试卤灵钠盐NSC 12097 sodium salt；试卤灵钠盐|||NSC 12097 sodium salt (2024/9/1)
简介：resorufin sodium salt (nsc-12097 sodium salt) is a fluorescent pink dye.
Resorufin；试卤灵NSC 12097；NSC 12097|||试卤灵 (2024/9/1)
简介：resorufin (nsc-12097) (nsc-12097) is a highly fluorescent pink dye.
Resolvin E1；化合物 T16733RvE1；RvE1 (2024/9/1)
简介：resolvin e1 is an effective endogenous pro-resolving mediator of inflammation. resolvin e1 has unique counterregulatory actions that inhibit pmn transendothelial migration. resolvin e1 also acts as an effective inhibitor of leukocyte infiltration, dendritic cell migration, and il-12 production.
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