9月
Rolziracetam；罗拉西坦CI-911；罗拉西坦|||CI-911 (2024/9/1)
简介：rolziracetam (ci-911) is a nootropic drug of the racetam family. it can improve short-term memory in rats and monkeys.
Rolofylline；洛罗茶碱KW-3902|||MK-7418|||KF-15372；KW-3902|||MK-7418|||KF-15372 (2024/9/1)
简介：rolofylline (kw-3902) is a selective adenosine a1 receptor antagonist used in the study of acute congestive heart failure and renal dysfunction, and in the study of neurodegenerative disorders.
Rogaratinib；化合物RogaratinibBAY1163877；BAY1163877 (2024/9/1)
简介：rogaratinib (bay1163877) is an aberrant inhibitor of fibroblast growth factor receptor (fgfr). rogaratinib is as an orally available, selective and potent inhibitor of fgfr-1, -2 and -3 kinase activity.
Rodatristat；化合物 T16780KAR5417；KAR5417 (2024/9/1)
简介：rodatristat is an effective tryptophan hydroxylase 1 and tph2 inhibitor (ic50s: 33 nm and 7 nm, respectively).
Nystatin；制霉菌素Stamycin|||Fungicidin|||Nystavescent；Stamycin|||Fungicidin|||制霉菌素|||Nystavescent (2024/9/1)
简介：nystatin (fungicidin) is a polyene antifungal antibiotic that is effective against yeast and mycoplasma and is orally active. nystatin can be used to treat skin and oropharyngeal candida infections.
Montelukast sodium孟鲁司特钠MK0476|||孟鲁司特钠 (2024/9/1)
简介：montelukast sodium (mk0476) is an orally available leukotriene receptor antagonist which is widely used for the prophylaxis and chronic treatment of asthma and has been linked to rare cases of clinically apparent liver injury.
Rodatristat ethyl；化合物RVT-014|||KAR5585|||RVT-1201；RVT-014|||KAR5585|||RVT-1201 (2024/9/1)
简介：rodatristat ethyl (kar5585) is a first-of-its-kind orally active and potent tryptophan hydroxylase 1 (tph1) inhibitor that significantly reduces 5-hydroxytryptamine (5-ht) levels and decreases pulmonary arterial hypertension (pah) at low concentrations.
Rocastine；罗卡斯汀AHR-11325；AHR-11325 (2024/9/1)
简介：rocastine (ahr-11325) is a selective and potent non-sedating h1 receptor antagonist.
ROC-325；化合物ROC-325ROC-325 (2024/9/1)
简介：roc-325 is an effective and orally active inhibitor of autophagy with anticancer activity. roc-325 induces renal cell carcinoma apoptosis and exhibits favorable selectivity.
RO9021；化合物RO9021RO9021 (2024/9/1)
简介：ro9021 is an orally bioavailable, novel atp-competitive syk inhibitor (average ic50: 5.6 nm).
Ro15-4513；化合物 T16775Ro15-4513 (2024/9/1)
简介：ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. ro15-4513 is an effective ethanol antagonist.
RO-9187；化合物 T16774RO-9187 (2024/9/1)
简介：ro-9187 is an effective hcv virus replication inhibitor(ic50: 171 nm).
Ro 90-7501化合物Ro 90-7501RO-90-7501 (2024/9/1)
简介：ro 90-7501 is an amyloid β42 (aβ42) protofibrillar and tpr-dependent pp5 inhibitor, a novel radiosensitiser for cervical cancer cells, which inhibits atm phosphorylation, promotes apoptosis, and induces cell-cycle arrest.ro 90-7501 exhibits antiviral activity and potential anticancer activity by inhibiting atm phosphorylation and dna repair, and by inhibiting hcmv.
Ro 64-6198；化合物 T16772Ro 64-6198 (2024/9/1)
简介：ro 64-6198 is a nonpeptide, high-affinity, and brain penetration n/ofq receptor (nop) agonist (ec50: 25.6 nm). ro 64-6198 is at least 100 times more selective for the nop receptor over the classic opioid receptors.
RO-5963；化合物RO-5963RO-5963 (2024/9/1)
简介：ro-5963 is a dual inhibitor of p53-mdm2 and p53-mdmx (ic50s: ~17 nm and ~24 nm, respectively).
Ro 41-1049 hydrochloride；化合物 T16770Ro 41-1049 hydrochloride (2024/9/1)
简介：ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine oxidase-a (kd: 16.5 and 64.4 nm, respectively).
Montelukast；孟鲁司特Singular；孟鲁司特|||Singular (2024/9/1)
简介：montelukast (singular) is an orally available leukotriene receptor antagonist which is widely used for the prophylaxis and chronic treatment of asthma and has been linked to rare cases of clinically apparent liver injury.
Ro 363；化合物 T16769Ro 363 (2024/9/1)
简介：ro 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contractility. ro 363 is an effective and highly selective β1-adrenoceptor agonist.
Ro-24-4736；化合物 T16768Ro-24-4736 (2024/9/1)
简介：ro 24-4736 is an effective and selective platelet-activating factor antagonist.
Ro-24-0238；化合物 T16767Ro-24-0238 (2024/9/1)
简介：ro-24-0238 is an antagonist of platelet-activating factor and inhibitor of thromboxane synthesis. ro-24-0238 used for lessening the inflammation and damage resulting from a local release of paf.
Ro 08-2750；化合物Ro 08-2750Ro 08-2750 (2024/9/1)
简介：ro 08-2750 is a non-peptide and reversible nerve growth factor (ngf) inhibitor which binds to ngf, and with an ic50 of ~ 1 µm. ro 08-2750 is a selective msi rna-binding activity inhibitor, with an ic50 of 2.7 μm. ro 08-2750 inhibits ngf binding to p75ntr selectively over trka.
RNPA1000；化合物 T16765RNPA1000 (2024/9/1)
简介：rnpa1000 is an attractive antimicrobial development candidate and rnpa inhibitor.
RN-18；化合物RN-18RN-18 (2024/9/1)
简介：rn-18 is an inhibitor of hiv-1 viral infectivity factor (ic50: 6 μm in nonpermissive h9 cells).
RN-1747；化合物RN-1747RN-1747 (2024/9/1)
简介：rn-1747 is a selective transient receptor potential cation channel subfamily v member 4 agonists (ec50: htrpv4 of 0.77 μm, mtrpv4 of 4.0 μm, and rtrpv4 of 4.1 μm). rn-1747 also antagonizes trpm8 (ic50: 4 μm).
RMC-4550；化合物RMC-4550RMC-4550 (2024/9/1)
简介：rmc-4550 is an effective and allosteric inhibitor of shp2 (ic50: 0.583 nm).
RK-287107；化合物RK-287107RK-287107 (2024/9/1)
简介：rk-287107 is an effective and specific inhibitor of tankyrase (ic50s: 14.3 and 10.6 nm for tankyrase-1 and tankyrase-2, respectively).
RK-24466；化合物RK-24466KIN 001-51；KIN 001-51 (2024/9/1)
简介：rk-24466 (kin 001-51) is a selective and potent inhibitor of lck, inhibits lck (64-509) and lckcd isoforms with ic50s of less than 1 and 2 nm, respectively.
Rosuvastatin；瑞舒伐他汀ZD 4522；罗伐他汀|||ZD 4522|||瑞舒伐他汀 (2024/9/1)
简介：rosuvastatin (zd 4522) is an antilipemic agent that competitively inhibits hydroxymethyl-glutaryl-coenzyme a (hmg-coa) reductase. hmg-coa reductase catalyzes the conversion of hmg-coa to mevalonic acid, the rate-limiting step in cholesterol biosynthesis. rosuvastatin belongs to a class of medications called statins and is used to reduce plasma cholesterol levels and prevent cardiovascular disease.
Ritanserin；利坦丝林R 55667；利坦丝林|||R 55667 (2024/9/1)
简介：ritanserin (r 55667) is a highly effective, relatively selective, long-acting antagonist of 5-ht2 receptor (ic50: 0.9 nm), less active on histamine h1, dopamine d2, adrenergic α1, adrenergic α2 receptors.
Rispenzepine；利喷西平Rispenzepine (2024/9/1)
简介：rispenzepine is a novel antagonist of muscarinic acetylcholine receptors (machrs), selectively targeting the m1 and m3 receptor subtypes, and can be used in the treatment of immune system disorders, infections, and respiratory diseases.
MSN交谈
