9月
RWJ-51204；化合物RWJ-51204RWJ-51204 (2024/9/1)
简介：rwj-51204 is a selective adenosine a2a receptor antagonist and a partial agonist of gaba(a) receptor (ic50: 0.2-2 nm). it has neuroprotective and movement-improving effects and can be used in research related to parkinson´s disease.
Ruzadolane；卢扎朵仑UP 26-91；卢扎朵仑|||UP 26-91 (2024/9/1)
简介：ruzadolane (formerly known as up 26-91) is a 5-hydroxytryptamine receptor antagonist developed as a non-narcotic central analgesic for the treatment of anxiety disorders and pain.
Aminophylline；氨茶碱Phyllocontin；氨茶碱|||Phyllocontin (2024/9/1)
简介：aminophylline (phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.
Rupintrivir芦平曲韦AG-7088|||AG7088|||Rupintrivirvr (2024/9/1)
简介：rupintrivirvr (ag7088) is a selective rhinovirus (hrv) 3c cysteine protease mimetic peptide inhibitor with antiviral and immunomodulatory activities.rupintrivirvr inhibits the replication of ev71 and ev-d68, and may be useful for the study of viral infections.
Runcaciguat；化合物RuncaciguatRuncaciguat (2024/9/1)
简介：runcaciguat is a soluble guanylate cyclase stimulator. runcaciguat combines with selective partial adenosine a1 receptor agonists and can be used in studies about cardiovascular and renal diseases.
Rucaparib monocamsylate；瑞卡帕布樟脑磺酸盐Rucaparib Camsylate；瑞卡帕布樟脑磺酸盐|||Rucaparib Camsylate (2024/9/1)
简介：rucaparib monocamsylate (rucaparib camsylate) is a parp inhibitor (parp1,ki of 1.4 nm). rucaparib camsylate also displays binding affinity to eight other parp domains.
RTS-V5；化合物 T16805RTS-V5 (2024/9/1)
简介：rts-v5 is a dual inhibitor of hdac/proteasome (ic50s: 6.9, 18, 15, 0.27, 0.53 μm for hdac1, hdac2, hdac3, hdac6, hdac8, respectively).
RS 8359；化合物RS 8359RS 8359 (2024/9/1)
简介：rs 8359 is a reversible inhibitor of monoamine oxidase a (mao-a) with a selectivity ratio of about 2200 for the a:b enzyme types. rs 8359 has antidepressant activity.
Lonapalene；氯萘帕林RS4317；RS4317 (2024/9/1)
简介：lonapalene (rs4317) is a 5-lipoxygenase (5-lo) inhibitor with anti-psoriasis efficacy.lonapalene topically blocks skin inflammation.
(RS)-(Tetrazol-5-yl)glycine；化合物(RS)-(Tetrazol-5-yl)glycineLY 285265|||D,L-(tetrazol-5-yl)glycine；LY (2024/9/1)
简介：(rs)-(tetrazol-5-yl)glycine (ly 285265) (d,l-(tetrazol-5-yl)glycine) is an effective and selective n-methyl-d-aspartate receptor agonist. (rs)-(tetrazol-5-yl)glycine has ec50s of 99 nm, 1.7 μm for glun1/glun2d, and glun1/glun2a, respectively.
(RS)-AMPA；化合物(RS)-AMPA(±)-AMPA；(±)-AMPA (2024/9/1)
简介：(rs)-ampa ((±)-ampa) is a glutamate analog. (rs)-ampa is an agonist of effective and selective excitatory neurotransmitter l-glutamic acid.
Tolazoline hydrochloride；苯甲唑啉盐酸盐Imidaline hydrochloride|||Imidaline (hydrochloride)|||Benzidazol hyd (2024/9/1)
简介：tolazoline hydrochloride (nsc35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn.
RS-246204；化合物 T16799RS-246204 (2024/9/1)
简介：rs-246204 is an r-spondin-1 substitute compound. rs-246204 is able to initiate small intestinal organoids without the use of the r-spondin-1 protein.
RS 17053 hydrochloride；化合物RS 17053 hydrochlorideRS-17053；RS-17053 (2024/9/1)
简介：rs 17053 hydrochloride is a potent and selective antagonist of α1a adrenoceptor. rs 17053 hydrochloride exhibits a pki value of 9.1 in native cell membrane and a pa2 value of 9.8 in functional assays.
RPR104632；化合物RPR104632RPR104632 (2024/9/1)
简介：rpr104632 is a novel and potent antagonist located at the nmda glycine site with neuroprotective activity.
RPR-260243；化合物 T16796RPR-260243 (2024/9/1)
简介：rpr-260243 is a novel activator of herg and modifies herg currents inhibited by dofetilide (ic50 = 58 nm).
Rpn11-IN-1；化合物 T16795Capzimin intermediate；Capzimin intermediate (2024/9/1)
简介：rpn11-in-1 is an effective and selective inhibitor of proteasome subunit rpn11 (ic50: 390 nm).
RO 4938581；化合物 T16794RO 4938581 (2024/9/1)
简介：ro 4938581 is an effective and selective agonist of gabaa α5 inverse (ki: 4.6 nm for gabaa α5β3γ2a, and shows a lower affinity at α1β3γ2a, α2β3γ2a, α3β3γ2a (ki, 174, 185, 80 nm, respectively)).
RO-28-1675；化合物 T16793Ro 28-1675；Ro 28-1675 (2024/9/1)
简介：ro 28-1675 is an effective allosteric gk activator (ic50: 0.24± 0.0019 um).
Rovazolac；化合物 RovazolacALX-101；ALX-101 (2024/9/1)
简介：rovazolac (alx-101) is a liver x receptor (lxr) modulator used in the study of immune system disorders and atopic dermatitis.
Rottlerin；粗糠柴苦素Mallotoxin|||NSC 56346|||NSC 94525；Mallotoxin|||NSC 56346|||粗糠柴苦素|||NSC 94525 (2024/9/1)
简介：rottlerin (nsc-56346) is a natural product purified from mallotus philippinensis and is a specific pkc inhibitor (ic50: pkcδ of 3-6 μm, pkcα,β,γ of 30-42 μm, pkcε,η,ζ of 80-100 μm). rottlerin causes apoptosis via caspase 3 activation.
Rotigaptide TFA(355151-12-1 free base)；化合物Rotigaptide TFARotigaptide TFA；Rotigaptide TFA (2024/9/1)
简介：rotigaptide tfa(355151-12-1 free base) is a novel and specific modulator of cx43 and is a potent aap. rotigaptide tfa(355151-12-1 free base) prevents the uncoupling of cx43-mediated gap junction communication and normalizes cell-to-cell communication during acute metabolic stress.
Rotigaptide；化合物 T16790ZP123；ZP123 (2024/9/1)
简介：rotigaptide is a novel and specific modulator of cx43 and is a potent aap. rotigaptide prevents the uncoupling of cx43-mediated gap junction communication and normalizes cell-to-cell communication during acute metabolic stress.
Thiostrepton；硫链丝菌素Thiactin|||Bryamycin|||Alaninamide；Thiactin|||Bryamycin|||Alaninamide|||硫链丝菌素 (2024/9/1)
简介：thiostrepton (alaninamide) is a one of the cyclic peptides from streptomyces that is active against gram-positive bacteria. in veterinary medicine, it has been used in mastitis caused by gram-negative organisms and in dermatologic disorders.
Rosoxacin；罗索沙星Acrosoxacin；罗索沙星|||Acrosoxacin (2024/9/1)
简介：rosoxacin (acrosoxacin) shows antibacterial activities against a broad spectrum of gram-negative bacteria including neisseria gonorrhoeae (mic90 = 0.03mg/ml).
Rosabulin；罗沙布林STA 5312；STA 5312 (2024/9/1)
简介：v rosabulin (sta 5312) is an orally active microtubule inhibitor with potency. rosabulin inhibits microtubule assembly and has broad-spectrum antitumor activity.
Vimirogant；化合物 T16787VTP-43742；VTP-43742 (2024/9/1)
简介：vimirogant is a rorγ inhibitor (ki: <100 nm).
Ropitoin；罗匹妥英TR 2985；罗匹妥英|||TR 2985 (2024/9/1)
简介：ropitoin is a novel drug of antiarrhythmics.
Ropidoxuridine；化合物RopidoxuridineIPdR；IPdR (2024/9/1)
简介：ropidoxuridine (ipdr) is a novel, orally available halogenated thymidine analogue that holds promise as a sensitizer for human tumors.ropidoxuridine is an orally available and bioavailable iudr (5-iodo-2´-deoxyuridine) prodrug.
Roniciclib；化合物RoniciclibBAY 1000394；BAY 1000394 (2024/9/1)
简介：roniciclib (bay 1000394) is a potent pan-cdk inhibitor and a novel oral cytotoxic agent. roniciclib inhibits the activity of cell-cycle cdks cdk1, cdk2, cdk3, cdk4, and of transcriptional cdks cdk7 and cdk9 with ic(50) values in the range between 5 and 25 nmol/l.
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