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(S)-Verapamil hydrochloride (S(-)-Verapamil hydrochloride) 通过 MRP1 抑制白三烯 C4 (LTC4) 和钙黄绿素的转运。(S)-Verapamil hydrochloride 导致潜在耐药性肿瘤细胞死亡。
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更新时间:2026/10/7 8:40:31关注度:2473
关键词标签:(S)-(-)-Verapamil,hydrochloride
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CAS No. : 36622-28-3
MCE 国际站:(S)-Verapamil hydrochloride
产品活性:(S)-Verapamil hydrochloride (S(-)-Verapamil hydrochloride) 通过 MRP1 抑制白三烯 C4 (LTC4) 和钙黄绿素的转运。(S)-Verapamil hydrochloride 导致潜在耐药性肿瘤细胞死亡。
研究领域:GPCR/G Protein | Neuronal Signaling | Membrane Transporter/Ion Channel | Apoptosis
作用靶点:Leukotriene Receptor | Calcium Channel | Apoptosis
In Vitro: (S)-Verapamil hydrochloride (S(-)-Verapamil hydrochloride) not the (R)-Verapamil hydrochloride potently induces the death of MRP1-transfected BHK-21 cells.
(S)-Verapamil hydrochloride is good active form and has the low bioavailability.
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