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Gluten Exorphin C

CAS No. : 142479-62⁻⁷

MCE 国际站：Gluten Exorphin C

产品活性：Gluten exorphin C 是一种源自谷朊粉的阿片肽。在 GPI 和 MVD 检测中，抑制 µ opioid 和 δ opioid 活性，IC₅₀ 值分别为 40 µM 和13.5 µM。

研究领域：GPCR/G Protein | Neuronal Signaling

作用靶点：Opioid Receptor

In Vitro: Gluten exorphin C, a novel opioid peptide, is isolated from the pepsin-trypsin-chymotrypsin digest of wheat gluten. Gluten exorphin C is evaluated its opioid activities by the GPI and MVD assays and its receptor affinities by radioreceptor assays. Its IC₅₀s are 40 µM and 13.5 µM in the GPI and the MVD assays, respectively. Gluten exorphin C has a structure quite different from any of the endogenous and exogenous opioid peptides ever reported in that the N terminal Tyr is the only aromatic amino acid. The analogs containing Tyr-Pro-X-Ser-Leu are synthesized to study its structure-activity relationship. Peptides in which X is an aromatic amino acid or an aliphatic hydrophobic amino acid has opioid activity.

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