MCE 的所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务。

[Leu5]-Enkephalin

CAS No. : 58822-25-6

MCE 国际站：[Leu5]-Enkephalin

产品活性：[Leu5]-Enkephalin 是一种具有吗啡药性的五肽。作为阿片受体 (opioid receptors) 激动剂。

研究领域：GPCR/G Protein | Neuronal Signaling | Metabolic Enzyme/Protease

作用靶点：Opioid Receptor | Endogenous Metabolite

In Vitro: Enkephalins (met- , leu-enkephalin, ａnd enkephalin 8) ａnd dynorphins are two classes of opioid peptides found in the spinal dorsal horn. Mu, delta, ａnd kappa are three major subtypes of opioid receptors. Enkephalins are putative endogenous ligands for delta opioid receptors, ａnd dynorphins are endogenous ligands for the kappa opioid receptors. Three receptor types resembling the vertebrate δ- ａnd κ-type opioid receptors have been characterized pharmacologically in nervous tissues (e.g. K_i=18.9 nM for Leu-enkephalin) ａnd localized by autoradiography at CHH terminals in the SG of C. maenas.Leucine-enkephalin is a pentapeptides with morphine like properties, naturally present in mammalian brain.

相关产品：Natural Product Library Plus | Bioactive Compound Library Plus | GPCR/G Protein Compound Library | Metabolism/Protease Compound Library | Neuronal Signaling Compound Library | Natural Product Library | Human Endogenous Metabolite Compound Library | Peptidomimetic Library | Neurotransmitter Receptor Compound Library | Rapamycin | 3-Methyladenine | Acetylcysteine | 5-Fluorouracil | ATP | Hydrocortisone | Retinoic acid | Docetaxel | Estradiol | Melatonin | Cytarabine | Nicotinamide | Isoprenaline hydrochloride | Prostaglandin E2 | Acetaminophen | (-)-Epigallocatechin Gallate | Calcitriol | β-Nicotinamide mononucleotide | DHEA | Liothyronine | Thymidine | NAD+ | Luteolin | Kaempferol | Cyclopamine | Genistein | Docosahexaenoic Acid | L-Glutathione reduced | Serotonin hydrochloride | Palmitic acid