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4(3H)-QuinazolinoneInhibitor,Bacterial,4(3H)-Quinazolinone,4(3H)Quinazolinone,inhibit,4(3H) Quinazol (2023/5/12)
简介：some 4-quinazolinone derivatives have antiplatelet activity.
CAY10594CAY10594,Inhibitor,CAY 10594,CAY-10594,Phospholipase,inhibit (2023/5/12)
简介：cay10594 is a potent phospholipase d2(pld2) inhibitor. cay10594 ameliorates acetaminophen-induced acute liver injury by regulating the phosphorylated-gsk-3β/jnk axis.
6-ChloropurineInhibitor,inhibit,6-Chloropurine,6Chloropurine,6 Chloropurine (2023/5/12)
简介：6-chloropurine is a building block in chemical synthesis,with antitumor activities.
CDN1163Inhibitor,CDN 1163,Calcium Channel,Ca channels,Ca2+ channels,CDN-1163,CDN1163,inhibit (2023/5/12)
简介：cdn1163 is a small molecule activator of sarco/endoplasmic reticulum ca2+-atpase (serca).
Procyanidin B3Histone Acetyltransferase,Procyanidin B-3,Procyanidin B 3,HAT,HATs,inhibit,Inhibitor,P (2023/5/12)
简介：procyanidin b3(b3) is a procyanidin dimer that is widely studied due to its high abundance in the human diet and antioxidant activity.
PLN-1474 (2023/5/12)
简介：pln-1474 is a potent αvβ1 inibitor with ic50 < 50nm (wo2021127483, compound 1)
CY5-SE Ditriethylamine salt (2023/5/12)
简介：cy5-se ditriethylamine salt is a reactive dye for the labeling of amino-groups in peptides, proteins, and oligonucleotides. excitation (nm):649, emission (nm): 670.
SR33805Ca channels,channel,failing,Ca2+ channels,Ca2+,SR 33805,Calcium Channel,acute,L-type,SR-33805 (2023/5/12)
简介：sr33805 is a potent antagonist of ca2+ channel(ec50s of 4.1 nm and 33 nm in depolarized and polarized conditions, respectively)
CycloleucineIonotropic glutamate receptors,inhibit,glycine,NMDA,cytostatic,nucleic,Inhibitor,Cyclole (2023/5/12)
简介：cycloleucine is an antagonist of nmda receptor associated glycine receptor with a ki of 600 μm. cycloleucine is also a competitive inhibitor of s-adenosyl-methionine mediated methylation with anxiolytic and cytostatic effects.
RLX-33 (2023/5/12)
简介：rlx-33 is a potent, selective and blood-brain barrier (bbb) penetrant antagonist of relaxin family peptide 3 (rxfp3, ic50=2.36 μm). rlx-33 also blocks relaxin-3-induced erk1/2 phosphorylation, with ic50s of 7.82 and 13.86 μm for erk1 and erk2 phosphorylation, respectively. rlx-33 can inhibits the stimulation of food intake induced by the rxfp3-selective agonist r3/i5 in rats.
Antimicrobial Compound 1Antimicrobial Compound 1 (2023/5/12)
简介：antimicrobial compound 1 is an alkyl pyridinium compound with tail 12c, head 4-carboxyl. antimicrobial compound 1 exhibits antimicrobial activities against b. subtilis and e. coli.
D18024D18024,D-18024 (2023/5/12)
简介：d18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.
1-ethyl-3-morpholin-4-yl-5,6,7,8-tetrahydroisoquinoline-4-carbonitrile (2023/5/12)
简介：1-ethyl-3-morpholin-4-yl-5,6,7,8-tetrahydroisoquinoline-4-carbonitrile is a positive allosteric modulator of mglur3 and can be used in studies about the treatment of parkinson´s disease.
1,3-DiphenylisobenzofuranROS,inhibit,oxygen,endoperoxide,1,3-Diphenylisobenzofuran,1,3Diphenylisoben (2023/5/12)
简介：1,3-diphenylisobenzofuran is a fluorescent probe. it possesses a highly specific reactivity towards singlet oxygen forming an endoperoxide which decomposes to give 1,2-dibenzoylbenzene. 1,3-diphenylisobenzofuran can detect the generation of reactive oxygen species (ros).
4i4i (2023/5/12)
简介：4i is a 5-ht3 receptor antagonist,it modulates the serotonergic system.
[Met5]-Enkephalin, amide TFA[Met5] Enkephalin, amide TFA,[Met-5]-Enkephalin, amide TFA,[Met5]Enkepha (2023/5/12)
简介：[met5]-enkephalin, amide tfa is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.
androsinInhibitor,inhibit,androsin (2023/5/12)
简介：androsin, isolated from picrorhiza kurroa royle ex benth, has anti-asthmatic effects.
4-Methylbenzylidene camphor4-Methylbenzylidene camphor,inhibit,Inhibitor,4 Methylbenzylidene camphor (2023/5/12)
简介：4-methylbenzylidene camphor is an ultraviolet light blocker used in cosmetics and sunscreen preparations ,specifically uv b radiation, also has estrogenic activities.
BAY-299 (2023/5/12)
简介：bay-299 is an effecitve inhibitor of the bromodomain and phd finger family member brpf2 and the tata box binding protein-associated factors taf1 and taf1l with ic50s of 67 nm, 8 nm, and 106 nm, respectively.
Farnesyl acetateFarnesyl acetate,inhibit,Farnesyl,Inhibitor (2023/5/12)
简介：farnesyl acetate is a flavouring compound identified in foods such as blueberries.
PBRM1-BD2-IN-5PBRM1BD2IN5 (2023/5/12)
简介：pbrm1-bd2-in-5 is a potent pbrm1 bromodomain inhibitor with kd values of 1.5 μm and 3.9 μm for pbrm1-bd2 and pbrm1-bd5, respectively, and an ic50 value of 0.26 μm for pbrm1-bd2. pbrm1-bd2-in-5 reduces the binding of full-length pbrm1 within the pbaf complex in cell lysates to acetylated histone peptide. pbrm1-bd2-in-5 can be used to research anticancer.
Quinizarincell,pesticide,Inhibitor,Quinizarin,DNA,Fungal,fungicide,DNA/RNA Synthesis,growth,tumor,in (2023/5/12)
简介：quinizarin is a natural product
SpinosinInhibitor,neuroprotective,Spinosin,inhibit,Aβ1-42 (2023/5/12)
简介：1. spinosin ameliorated memory impairment induced through aβo, the serotonergic neurotransmitter system, and these effects were regulated, in part, through neuroprotective activity via the anti-inflammatory effects of spinosin. 2. spinosin exerts anxiolytic-like effects, and its mechanism of action appears to be modulated by gabaa and 5-ht1a receptors. 3. there was a wide brain regional tissue distribution of spinosin. the concentrations of spinosin in corpus striatum and hippocampus were higher
Thyrotropin-Releasing Hormone (TRH), Free AcidThyrotropin Releasing Hormone (TRH), Free Acid,inhibit (2023/5/12)
简介：thyrotropin-releasing hormone (trh), free acid (trh-oh) causes a variety of thyroidal and non-thyroidal effects, the best known being the feedback regulation of thyroid hormone levels.
N,N-Bis(2-hydroxyethyl)-p-phenylenediamiN,NBis(2hydroxyethyl)pphenylenediami,N,N Bis(2 hydroxyethyl) (2023/5/12)
简介：
Hydroxyprogesterone caproateHydroxyprogesterone caproate,Inhibitor,inhibit (2023/5/12)
简介：hydroxyprogesterone caproate is a synthetic progestational agent. it binds to and activates nuclear progesterone receptors in the reproductive system and inhibits ovulation and an alteration in the cervical mucus and endometrium.
Naphthol AS-EHAT,KIX-KID,MCF-7,cancer,Inhibitor,Naphthol AS-E,inhibit,Epigenetic Reader Domain,CREB, (2023/5/12)
简介：nas-e is an the kix-kid interaction and creb-mediated gene transcription inhibitor.
ParicalcitolVitamin D receptor,Paricalcitol,Vitamin D,Inhibitor,VD/VDR,inhibit (2023/5/12)
简介：paricalcitol is a vitamin d receptor agonist. it is used for the prevention and treatment of secondary hyperparathyroidism associated with chronic renal failure.
NSC348884lymphoma,cancer,inhibit,SKOV3,MOSEC/Luc cell,NSC-348884,NSC 348884,LNCaP,doxorubicin,NSC348 (2023/5/12)
简介：nsc348884 is a nucleophosmin inhibitor disrupts oligomer formation and induces apoptosis, inhibits cell proliferation at an ic50 of 1.7-4.0 μm in distinct cancer cell lines.
ASK1-IN-2colitis,ulcerative,signal-regulating,ASK1 IN 2,ASK1IN2,inhibit,MAP kinase kinase kinase, ME (2023/5/12)
简介：ask1-in-2 is a potent and orally active inhibitor of apoptosis signal-regulating kinase 1 (ask1), with an ic50 of 32.8 nm. ask1-in-2 can potentially be used as a therapeutic strategy for ulcerative colitis[1].
MSN交谈
